Synthesis of Islatravir Enabled by a Catalytic, Enantioselective Alkynylation of a Ketone.
Patel NR, Nawrat CC, McLaughlin M, Xu Y, Huffman MA, Yang H, Li H, Whittaker AM, Andreani T, Lévesque F, Fryszkowska A, Brunskill A, Tschaen DM, Maloney KM.
Patel NR, et al. Among authors: huffman ma.
Org Lett. 2020 Jun 19;22(12):4659-4664. doi: 10.1021/acs.orglett.0c01431. Epub 2020 Jun 9.
Org Lett. 2020.
PMID: 32516536