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Page 1
Oxamides as novel NR2B selective NMDA receptor antagonists.
Barta-Szalai G, Borza I, Bozó E, Kiss C, Agai B, Proszenyák A, Keseru GM, Gere A, Kolok S, Galgóczy K, Horváth C, Farkas S, Domány G. Barta-Szalai G, et al. Among authors: bozo e. Bioorg Med Chem Lett. 2004 Aug 2;14(15):3953-6. doi: 10.1016/j.bmcl.2004.05.053. Bioorg Med Chem Lett. 2004. PMID: 15225705
Indole-2-carboxamides as novel NR2B selective NMDA receptor antagonists.
Borza I, Kolok S, Gere A, Agai-Csongor E, Agai B, Tárkányi G, Horváth C, Barta-Szalai G, Bozó E, Kiss C, Bielik A, Nagy J, Farkas S, Domány G. Borza I, et al. Among authors: bozo e. Bioorg Med Chem Lett. 2003 Nov 3;13(21):3859-61. doi: 10.1016/s0960-894x(03)00708-x. Bioorg Med Chem Lett. 2003. PMID: 14552795
Selective NR1/2B N-methyl-D-aspartate receptor antagonists among indole-2-carboxamides and benzimidazole-2-carboxamides.
Borza I, Bozó E, Barta-Szalai G, Kiss C, Tárkányi G, Demeter A, Gáti T, Háda V, Kolok S, Gere A, Fodor L, Nagy J, Galgóczy K, Magdó I, Agai B, Fetter J, Bertha F, Keserü GM, Horváth C, Farkas S, Greiner I, Domány G. Borza I, et al. Among authors: bozo e. J Med Chem. 2007 Mar 8;50(5):901-14. doi: 10.1021/jm060420k. Epub 2007 Feb 10. J Med Chem. 2007. PMID: 17290978
Quinolinyl- and phenantridinyl-acetamides as bradykinin B1 receptor antagonists.
Eles J, Beke G, Vágó I, Bozó E, Huszár J, Tarcsay A, Kolok S, Schmidt E, Vastag M, Hornok K, Farkas S, Domány G, Keserű GM. Eles J, et al. Among authors: bozo e. Bioorg Med Chem Lett. 2012 May 1;22(9):3095-9. doi: 10.1016/j.bmcl.2012.03.065. Epub 2012 Mar 21. Bioorg Med Chem Lett. 2012. PMID: 22483585
Discovery of novel positive allosteric modulators of the α7 nicotinic acetylcholine receptor: Scaffold hopping approach.
Ledneczki I, Tapolcsányi P, Gábor E, Visegrády A, Vass M, Éles J, Holm P, Horváth A, Pocsai A, Mahó S, Greiner I, Krámos B, Béni Z, Kóti J, Káncz AE, Thán M, Kolok S, Laszy J, Balázs O, Bugovits G, Nagy J, Vastag M, Szájli Á, Bozó É, Lévay G, Lendvai B, Némethy Z. Ledneczki I, et al. Among authors: bozo e. Eur J Med Chem. 2021 Mar 15;214:113189. doi: 10.1016/j.ejmech.2021.113189. Epub 2021 Jan 14. Eur J Med Chem. 2021. PMID: 33540354
Synthesis and Characterization of New V1A Antagonist Compounds: The Separation of Four Atropisomeric Stereoisomers.
Szeleczky Z, Szakács Z, Bozó É, Baska F, Vukics K, Lévai S, Temesvári K, Vass E, Béni Z, Krámos B, Magdó I, Szántay C Jr, Kóti J, Domány-Kovács K, Greiner I, Bata I. Szeleczky Z, et al. Among authors: bozo e. J Med Chem. 2021 Jul 22;64(14):10445-10468. doi: 10.1021/acs.jmedchem.1c00863. Epub 2021 Jul 13. J Med Chem. 2021. PMID: 34255509
Discovery and Characterization of RGH-122, a Potent, Selective, and Orally Bioavailable V1a Receptor Antagonist.
Baska F, Bozó É, Szeleczky Z, Szántó G, Vukics K, Szakács Z, Domány-Kovács K, Kurkó D, Vass E, Thán M, Vastag M, Temesvári K, Lévai S, Halász AS, Szondiné Kordás K, Román V, Greiner I, Bata I. Baska F, et al. Among authors: bozo e. J Med Chem. 2024 Jan 11;67(1):643-673. doi: 10.1021/acs.jmedchem.3c01868. Epub 2024 Jan 2. J Med Chem. 2024. PMID: 38165765
31 results