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Novel heteroarotinoids as potential antagonists of Mycobacterium bovis BCG.
J Med Chem. 2004 Feb 12;47(4):1008-17. doi: 10.1021/jm0303453.
J Med Chem. 2004.
PMID: 14761203
Synthesis, structure-activity relationships, and RARgamma-ligand interactions of nitrogen heteroarotinoids.
Dhar A, Liu S, Klucik J, Berlin KD, Madler MM, Lu S, Ivey RT, Zacheis D, Brown CW, Nelson EC, Birckbichler PJ, Benbrook DM.
Dhar A, et al. Among authors: klucik j.
J Med Chem. 1999 Sep 9;42(18):3602-14. doi: 10.1021/jm9900974.
J Med Chem. 1999.
PMID: 10479291
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Heteroarotinoids inhibit head and neck cancer cell lines in vitro and in vivo through both RAR and RXR retinoic acid receptors.
Zacheis D, Dhar A, Lu S, Madler MM, Klucik J, Brown CW, Liu S, Clement F, Subramanian S, Weerasekare GM, Berlin KD, Gold MA, Houck JR Jr, Fountain KR, Benbrook DM.
Zacheis D, et al. Among authors: klucik j.
J Med Chem. 1999 Oct 21;42(21):4434-45. doi: 10.1021/jm990292i.
J Med Chem. 1999.
PMID: 10543887
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Synthesis, structure-activity relationships, and RARgamma-ligand interactions of nitrogen heteroarotinoids.
Dhar A, Liu S, Klucik J, Berlin KD, Madler MM, Lu S, Ivey RT, Zacheis D, Brown CW, Nelson EC, Birckbichler PJ, Benbrook DM.
Dhar A, et al. Among authors: klucik j.
J Med Chem. 2000 Jan 27;43(2):303. doi: 10.1021/jm990593s.
J Med Chem. 2000.
PMID: 10650065
No abstract available.
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2-(Arylmethyl)-3-substituted quinuclidines as selective alpha 7 nicotinic receptor ligands.
Mazurov A, Klucik J, Miao L, Phillips TY, Seamans A, Schmitt JD, Hauser TA, Johnson RT Jr, Miller C.
Mazurov A, et al. Among authors: klucik j.
Bioorg Med Chem Lett. 2005 Apr 15;15(8):2073-7. doi: 10.1016/j.bmcl.2005.02.045.
Bioorg Med Chem Lett. 2005.
PMID: 15808471
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Synthesis of ent-kaurane diterpene monoglycosides.
Chaturvedula VS, Klucik J, Upreti M, Prakash I.
Chaturvedula VS, et al. Among authors: klucik j.
Molecules. 2011 Oct 3;16(10):8402-9. doi: 10.3390/molecules16108402.
Molecules. 2011.
PMID: 21968534
Free PMC article.
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Targacept active conformation search: a new method for predicting the conformation of a ligand bound to its protein target.
Klucik J, Xiao YD, Hammond PS, Harris R, Schmitt JD.
Klucik J, et al.
J Med Chem. 2004 Dec 30;47(27):6831-9. doi: 10.1021/jm049729z.
J Med Chem. 2004.
PMID: 15615532
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