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Novel piperidinium and pyridinium agents as water-soluble acetylcholinesterase inhibitors for the reversal of neuromuscular blockade.
Bioorg Med Chem Lett. 2002 Sep 16;12(18):2569-72. doi: 10.1016/s0960-894x(02)00483-3.
Bioorg Med Chem Lett. 2002.
PMID: 12182862
Quaternary salts of E2020 analogues as acetylcholinesterase inhibitors for the reversal of neuromuscular block.
Clark JK, Cowley P, Muir AW, Palin R, Pow E, Prosser AB, Taylor R, Zhang MQ.
Clark JK, et al. Among authors: prosser ab.
Bioorg Med Chem Lett. 2002 Sep 16;12(18):2565-8. doi: 10.1016/s0960-894x(02)00482-1.
Bioorg Med Chem Lett. 2002.
PMID: 12182861
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Cyclodextrin-derived host molecules as reversal agents for the neuromuscular blocker rocuronium bromide: synthesis and structure-activity relationships.
Adam JM, Bennett DJ, Bom A, Clark JK, Feilden H, Hutchinson EJ, Palin R, Prosser A, Rees DC, Rosair GM, Stevenson D, Tarver GJ, Zhang MQ.
Adam JM, et al.
J Med Chem. 2002 Apr 25;45(9):1806-16. doi: 10.1021/jm011107f.
J Med Chem. 2002.
PMID: 11960492
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Structure-activity relationships and CoMFA of N-3 substituted phenoxypropyl piperidine benzimidazol-2-one analogues as NOP receptor agonists with analgesic properties.
Palin R, Clark JK, Evans L, Houghton AK, Jones PS, Prosser A, Wishart G, Yoshiizumi K.
Palin R, et al.
Bioorg Med Chem. 2008 Mar 15;16(6):2829-51. doi: 10.1016/j.bmc.2008.01.005. Epub 2008 Jan 10.
Bioorg Med Chem. 2008.
PMID: 18249547
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The discovery of novel indole-2-carboxamides as cannabinoid CB(1) receptor antagonists.
Cowley PM, Baker J, Barn DR, Buchanan KI, Carlyle I, Clark JK, Clarkson TR, Deehan M, Edwards D, Goodwin RR, Jaap D, Kiyoi Y, Mort C, Palin R, Prosser A, Walker G, Ward N, Wishart G, Young T.
Cowley PM, et al.
Bioorg Med Chem Lett. 2011 Jan 1;21(1):497-501. doi: 10.1016/j.bmcl.2010.10.104. Epub 2010 Oct 26.
Bioorg Med Chem Lett. 2011.
PMID: 21075628
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Discovery of potent and orally bioavailable heterocycle-based cannabinoid CB1 receptor agonists.
Kiyoi T, Adam JM, Clark JK, Davies K, Easson AM, Edwards D, Feilden H, Fields R, Francis S, Jeremiah F, McArthur D, Morrison AJ, Prosser A, Ratcliffe PD, Schulz J, Wishart G, Baker J, Campbell R, Cottney JE, Deehan M, Epemolu O, Evans L.
Kiyoi T, et al.
Bioorg Med Chem Lett. 2011 Mar 15;21(6):1748-53. doi: 10.1016/j.bmcl.2011.01.082. Epub 2011 Jan 22.
Bioorg Med Chem Lett. 2011.
PMID: 21316962
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Low brain penetrant CB1 receptor agonists for the treatment of neuropathic pain.
Adam JM, Clark JK, Davies K, Everett K, Fields R, Francis S, Jeremiah F, Kiyoi T, Maidment M, Morrison A, Ratcliffe P, Prosser A, Schulz J, Wishart G, Baker J, Boyce S, Campbell R, Cottney JE, Deehan M, Martin I.
Adam JM, et al.
Bioorg Med Chem Lett. 2012 Apr 15;22(8):2932-7. doi: 10.1016/j.bmcl.2012.02.048. Epub 2012 Feb 23.
Bioorg Med Chem Lett. 2012.
PMID: 22421020
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