Gao LJ - Search Results

1

Synthesis and affinity studies of himbacine derived muscarinic receptor antagonists.

Gao LJ, Waelbroeck M, Hofman S, Van Haver D, Milanesio M, Viterbo D, De Clercq PJ. Gao LJ, et al. Bioorg Med Chem Lett. 2002 Aug 5;12(15):1909-12. doi: 10.1016/s0960-894x(02)00315-3. Bioorg Med Chem Lett. 2002. PMID: 12113806

2

A novel short convergent entry into himbacine derivatives.

Van Cauwenberge G, Gao LJ, Van Haver D, Milanesio M, Viterbo D, De Clercq PJ. Van Cauwenberge G, et al. Among authors: gao lj. Org Lett. 2002 May 2;4(9):1579-82. doi: 10.1021/ol025801g. Org Lett. 2002. PMID: 11975633

3

Previtamin D3 with a trans-fused decalin CD-ring has pronounced genomic activity.

Verlinden L, Verstuyf A, Verboven C, Eelen G, De Ranter C, Gao LJ, Chen YJ, Murad I, Choi M, Yamamoto K, Yamada S, Van Haver D, Vandewalle M, De Clercq PJ, Bouillon R. Verlinden L, et al. Among authors: gao lj. J Biol Chem. 2003 Sep 12;278(37):35476-82. doi: 10.1074/jbc.M302045200. Epub 2003 Jun 26. J Biol Chem. 2003. PMID: 12829710 Free article.

4

Synthesis, biological activity, and conformational analysis of CD-ring modified trans-decalin 1 alpha,25-dihydroxyvitamin D analogs.

Chen YJ, Gao LJ, Murad I, Verstuyf A, Verlinden L, Verboven C, Bouillon R, Viterbo D, Milanesio M, Van Haver D, Vandewalle M, De Clercq PJ. Chen YJ, et al. Among authors: gao lj. Org Biomol Chem. 2003 Jan 21;1(2):257-67. doi: 10.1039/b209147j. Org Biomol Chem. 2003. PMID: 12929421

5

Biological activity and conformational analysis of C20 and C14 epimers of CD-ring modified trans-decalin 1alpha,25-dihydroxyvitamin D analogs.

De Clercq PJ, Murad I, Gao LJ, Chen YJ, Van Haver D, Vandewalle M, Verstuyf A, Verlinden L, Verboven C, Bouillon R. De Clercq PJ, et al. Among authors: gao lj. J Steroid Biochem Mol Biol. 2004 May;89-90(1-5):61-6. doi: 10.1016/j.jsbmb.2004.03.052. J Steroid Biochem Mol Biol. 2004. PMID: 15225748

6

Synthesis and in vitro evaluation of 2-amino-4-N-piperazinyl-6-(3,4-dimethoxyphenyl)-pteridines as dual immunosuppressive and anti-inflammatory agents.

De Jonghe S, Marchand A, Gao LJ, Calleja A, Cuveliers E, Sienaert I, Herman J, Clydesdale G, Sefrioui H, Lin Y, Pfleiderer W, Waer M, Herdewijn P. De Jonghe S, et al. Among authors: gao lj. Bioorg Med Chem Lett. 2011 Jan 1;21(1):145-9. doi: 10.1016/j.bmcl.2010.11.053. Epub 2010 Nov 16. Bioorg Med Chem Lett. 2011. PMID: 21131199 Free article.

7

Synthesis and evaluation of novel ligands for the histamine H₄ receptor based on a pyrrolo[2,3-d]pyrimidine scaffold.

Gao LJ, Schwed JS, Weizel L, De Jonghe S, Stark H, Herdewijn P. Gao LJ, et al. Bioorg Med Chem Lett. 2013 Jan 1;23(1):132-7. doi: 10.1016/j.bmcl.2012.10.139. Epub 2012 Nov 15. Bioorg Med Chem Lett. 2013. PMID: 23218604

8

Discovery of dual death-associated protein related apoptosis inducing protein kinase 1 and 2 inhibitors by a scaffold hopping approach.

Gao LJ, Kovackova S, Sála M, Ramadori AT, De Jonghe S, Herdewijn P. Gao LJ, et al. J Med Chem. 2014 Sep 25;57(18):7624-43. doi: 10.1021/jm5007929. Epub 2014 Sep 11. J Med Chem. 2014. PMID: 25178155

9

Discovery of 7-N-piperazinylthiazolo[5,4-d]pyrimidine analogues as a novel class of immunosuppressive agents with in vivo biological activity.

Jang MY, Lin Y, De Jonghe S, Gao LJ, Vanderhoydonck B, Froeyen M, Rozenski J, Herman J, Louat T, Van Belle K, Waer M, Herdewijn P. Jang MY, et al. Among authors: gao lj. J Med Chem. 2011 Jan 27;54(2):655-68. doi: 10.1021/jm101254z. Epub 2010 Dec 20. J Med Chem. 2011. PMID: 21171614

10

Synthesis and structure-activity relationship studies of 2-(1,3,4-oxadiazole-2(3H)-thione)-3-amino-5-arylthieno[2,3-b]pyridines as inhibitors of DRAK2.

Leonczak P, Gao LJ, Ramadori AT, Lescrinier E, Rozenski J, De Jonghe S, Herdewijn P. Leonczak P, et al. Among authors: gao lj. ChemMedChem. 2014 Nov;9(11):2587-601. doi: 10.1002/cmdc.201402234. Epub 2014 Aug 21. ChemMedChem. 2014. PMID: 25146684

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