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Aminoglycoside-modifying enzymes: mechanisms of catalytic processes and inhibition.
Drug Resist Updat. 2001 Apr;4(2):106-17. doi: 10.1054/drup.2001.0197.
Drug Resist Updat. 2001.
PMID: 11512519
Review.
Aminoglycosides modified by resistance enzymes display diminished binding to the bacterial ribosomal aminoacyl-tRNA site.
Llano-Sotelo B, Azucena EF Jr, Kotra LP, Mobashery S, Chow CS.
Llano-Sotelo B, et al. Among authors: azucena ef jr.
Chem Biol. 2002 Apr;9(4):455-63. doi: 10.1016/s1074-5521(02)00125-4.
Chem Biol. 2002.
PMID: 11983334
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Tethered bisubstrate derivatives as probes for mechanism and as inhibitors of aminoglycoside 3'-phosphotransferases.
Liu M, Haddad J, Azucena E, Kotra LP, Kirzhner M, Mobashery S.
Liu M, et al. Among authors: azucena e.
J Org Chem. 2000 Nov 3;65(22):7422-31. doi: 10.1021/jo000589k.
J Org Chem. 2000.
PMID: 11076599
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Design of novel antibiotics that bind to the ribosomal acyltransfer site.
Haddad J, Kotra LP, Llano-Sotelo B, Kim C, Azucena EF Jr, Liu M, Vakulenko SB, Chow CS, Mobashery S.
Haddad J, et al. Among authors: azucena ef jr.
J Am Chem Soc. 2002 Apr 3;124(13):3229-37. doi: 10.1021/ja011695m.
J Am Chem Soc. 2002.
PMID: 11916405
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The SRC substrate Tks5, podosomes (invadopodia), and cancer cell invasion.
Courtneidge SA, Azucena EF, Pass I, Seals DF, Tesfay L.
Courtneidge SA, et al. Among authors: azucena ef.
Cold Spring Harb Symp Quant Biol. 2005;70:167-71. doi: 10.1101/sqb.2005.70.014.
Cold Spring Harb Symp Quant Biol. 2005.
PMID: 16869750
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The adaptor protein Tks5/Fish is required for podosome formation and function, and for the protease-driven invasion of cancer cells.
Seals DF, Azucena EF Jr, Pass I, Tesfay L, Gordon R, Woodrow M, Resau JH, Courtneidge SA.
Seals DF, et al. Among authors: azucena ef jr.
Cancer Cell. 2005 Feb;7(2):155-65. doi: 10.1016/j.ccr.2005.01.006.
Cancer Cell. 2005.
PMID: 15710328
Free article.
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