Tiotidine, a classical H2-antagonist, presents characteristics of an inverse agonist in U937 cell line

Inflamm Res. 1998:47 Suppl 1:S42-3. doi: 10.1007/s000110050260.
No abstract available

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Cimetidine / analogs & derivatives*
  • Cimetidine / pharmacology
  • Cyclic AMP / analysis
  • Cyclic AMP / metabolism
  • Dose-Response Relationship, Drug
  • Guanidines / pharmacology
  • Histamine Agonists / pharmacology
  • Histamine H2 Antagonists / pharmacology*
  • Humans
  • Imidazoles / pharmacology
  • Lymphoma, Large B-Cell, Diffuse
  • Receptors, Histamine H2 / classification
  • Receptors, Histamine H2 / drug effects
  • Tumor Cells, Cultured

Substances

  • Guanidines
  • Histamine Agonists
  • Histamine H2 Antagonists
  • Imidazoles
  • Receptors, Histamine H2
  • BU-E 75
  • Cimetidine
  • Cyclic AMP
  • tiotidine