Inhibition of terfenadine metabolism. Pharmacokinetic and pharmacodynamic consequences

Clin Pharmacokinet. 1994 Jul;27(1):1-5. doi: 10.2165/00003088-199427010-00001.
No abstract available

Publication types

  • Research Support, Non-U.S. Gov't
  • Review

MeSH terms

  • Cytochrome P-450 Enzyme System / metabolism
  • Drug Interactions
  • Fluconazole / pharmacology*
  • Heart / drug effects
  • Humans
  • Itraconazole / pharmacology*
  • Ketoconazole / pharmacology*
  • Prodrugs / adverse effects
  • Prodrugs / pharmacokinetics*
  • Terfenadine / adverse effects
  • Terfenadine / antagonists & inhibitors
  • Terfenadine / pharmacokinetics*

Substances

  • Prodrugs
  • Itraconazole
  • Terfenadine
  • Fluconazole
  • Cytochrome P-450 Enzyme System
  • Ketoconazole