Receptor binding properties of four-helix-bundle growth factors deduced from electrostatic analysis

Protein Sci. 1994 Jun;3(6):920-35. doi: 10.1002/pro.5560030607.

Abstract

Hormones of the hematopoietin class mediate signal transduction by binding to specific transmembrane receptors. Structural data show that the human growth hormone (hGH) forms a complex with a homodimeric receptor and that hGH is a member of a class of hematopoietins possessing an antiparallel 4-alpha-helix bundle fold. Mutagenesis experiments suggest that electrostatic interactions may have an important influence on hormone-receptor recognition. In order to examine the specificity of hormone-receptor complexation, an analysis was made of the electrostatic potentials of hGH, interleukin-2 (IL-2), interleukin-4 (IL-4), granulocyte colony-stimulating factor (G-CSF), granulocyte-macrophage colony-stimulating factor (GM-CSF), and the hGH and IL-4 receptors. The binding surfaces of hGH and its receptor, and of IL-4 and its receptor, show complementary electrostatic potentials. The potentials of the hGH and its receptor display approximately 2-fold rotational symmetry because the receptor subunits are identical. In contrast, the potentials of GM-CSF and IL-2 lack such symmetry, consistent with their known high affinity for hetero-oligomeric receptors. Analysis of the electrostatic potentials supports a recently proposed hetero-oligomeric model for a high-affinity IL-4 receptor and suggests a possible new receptor binding mode for G-CSF; it also provides valuable information for guiding structural and mutagenesis studies of signal-transducing proteins and their receptors.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Electrochemistry
  • Granulocyte Colony-Stimulating Factor / chemistry
  • Granulocyte-Macrophage Colony-Stimulating Factor / chemistry
  • Growth Hormone / chemistry
  • Growth Hormone / metabolism
  • Growth Substances / chemistry*
  • Growth Substances / metabolism*
  • Humans
  • Interleukin-2
  • Interleukin-4
  • Macromolecular Substances
  • Magnetic Resonance Spectroscopy
  • Models, Molecular
  • Protein Structure, Secondary*
  • Receptors, Growth Factor / chemistry
  • Receptors, Growth Factor / metabolism*
  • Receptors, Interleukin-4
  • Receptors, Mitogen / chemistry
  • Receptors, Mitogen / metabolism
  • Receptors, Somatotropin / chemistry
  • Receptors, Somatotropin / metabolism

Substances

  • Growth Substances
  • Interleukin-2
  • Macromolecular Substances
  • Receptors, Growth Factor
  • Receptors, Interleukin-4
  • Receptors, Mitogen
  • Receptors, Somatotropin
  • Granulocyte Colony-Stimulating Factor
  • Interleukin-4
  • Granulocyte-Macrophage Colony-Stimulating Factor
  • Growth Hormone