No abstract available
Keywords:
ADME/Tox; drug design; in vitro assays; molecular chameleon; oral druggable space.
MeSH terms
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Administration, Oral
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Biological Availability
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Cell Membrane / drug effects
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Enzyme Inhibitors / administration & dosage
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Enzyme Inhibitors / chemistry
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Enzyme Inhibitors / pharmacokinetics*
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Humans
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Ligands
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Molecular Structure
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Permeability / drug effects
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Proteolysis / drug effects
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Ubiquitin-Protein Ligases / antagonists & inhibitors*
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Ubiquitin-Protein Ligases / metabolism
Substances
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Enzyme Inhibitors
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Ligands
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Ubiquitin-Protein Ligases