No abstract available
Keywords:
DPAGT1; anticancer drugs; co-crystal structures; inhibitors; structure-based drug design.
Publication types
-
Editorial
-
Research Support, N.I.H., Extramural
-
Research Support, Non-U.S. Gov't
MeSH terms
-
Animals
-
Biosynthetic Pathways / drug effects
-
Drug Design*
-
Drug Discovery
-
Enzyme Inhibitors / chemistry
-
Enzyme Inhibitors / pharmacology*
-
Humans
-
Molecular Docking Simulation
-
N-Acetylglucosaminyltransferases / antagonists & inhibitors*
-
N-Acetylglucosaminyltransferases / chemistry
-
N-Acetylglucosaminyltransferases / metabolism
-
Polysaccharides / metabolism*
Substances
-
Enzyme Inhibitors
-
Polysaccharides
-
N-Acetylglucosaminyltransferases
-
dolichyl-phosphate alpha-N-acetylglucosaminyltransferase