MEP50/PRMT5-mediated methylation activates GLI1 in Hedgehog signalling through inhibition of ubiquitination by the ITCH/NUMB complex

Commun Biol. 2019 Jan 18:2:23. doi: 10.1038/s42003-018-0275-4. eCollection 2019.

Abstract

Transcription factor GLI1 is an effecter of Hedgehog (HH) signalling and activated in a broad spectrum of cancers. However, the role of the HH-GLI1 pathway in cancer and the activation mechanism of GLI1 in HH signalling after dissociation from its inhibitor, SUFU, are not fully understood. Here, we found that GLI1 associated with the methylosome protein 50 (MEP50)/protein arginine methyltransferase 5 (PRMT5) complex and was methylated. Association of MEP50/PRMT5 with GLI1 was enhanced and expression of MEP50 and PRMT5 was activated by HH signals, suggesting their role in positive feedback regulation. Methylated GLI1 lost its ability to bind ubiquitin ligase ITCH/NUMB, resulting in nuclear accumulation and activation of GLI1. Moreover, protein expression of GLI1 was enhanced by MEP50/PRMT5 and expression of MEP50, PRMT5, and GLI1 target genes was upregulated in HH-expressing cancers. These results suggest that MEP50/PRMT5 is important for HH signal-induced GLI1 activation, especially in cancers.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Adaptor Proteins, Signal Transducing / metabolism*
  • Cell Line
  • Hedgehog Proteins / metabolism*
  • Humans
  • Membrane Proteins / metabolism*
  • Methylation
  • Models, Biological
  • Multiprotein Complexes
  • Nerve Tissue Proteins / metabolism*
  • Protein Binding
  • Protein-Arginine N-Methyltransferases / metabolism*
  • Repressor Proteins / metabolism*
  • Signal Transduction*
  • Ubiquitin-Protein Ligases / metabolism*
  • Ubiquitination
  • Zinc Finger Protein GLI1 / metabolism*

Substances

  • Adaptor Proteins, Signal Transducing
  • GLI1 protein, human
  • Hedgehog Proteins
  • MEP50 protein, human
  • Membrane Proteins
  • Multiprotein Complexes
  • Nerve Tissue Proteins
  • NUMB protein, human
  • Repressor Proteins
  • Zinc Finger Protein GLI1
  • PRMT5 protein, human
  • Protein-Arginine N-Methyltransferases
  • ITCH protein, human
  • Ubiquitin-Protein Ligases