Development of injectable liposomes and drug-in-cyclodextrin-in-liposome formulations encapsulating estetrol to prevent cerebral ischemia of premature babies

Eur J Pharm Sci. 2019 Jan 15:127:52-59. doi: 10.1016/j.ejps.2018.10.006. Epub 2018 Oct 9.
No abstract available

Keywords: Blood-brain barrier; Cerebral ischemia; Drug-in-Cyclodextrin-in-liposome; Estetrol; Hemocompatibility; Liposome.

MeSH terms

  • Biocompatible Materials / chemistry
  • Blood-Brain Barrier / metabolism
  • Brain Ischemia / prevention & control*
  • Cell Survival / drug effects
  • Cells, Cultured
  • Cyclodextrins / chemistry*
  • Drug Compounding
  • Drug Liberation
  • Drug Stability
  • Estetrol / administration & dosage
  • Estetrol / pharmacology*
  • Humans
  • Infant, Newborn
  • Infant, Premature
  • Liposomes / chemistry*
  • Particle Size
  • Permeability
  • Surface Properties
  • Thrombin / metabolism

Substances

  • Biocompatible Materials
  • Cyclodextrins
  • Liposomes
  • Thrombin
  • Estetrol