Histone acetyltransferase inhibitors: where art thou?

Future Med Chem. 2016 Sep;8(13):1525-8. doi: 10.4155/fmc-2016-0151. Epub 2016 Aug 24.

Authors

Jonathan B Baell¹, Wenjun Miao²

Affiliations

¹ Medicinal Chemistry, Monash Institute of Pharmaceutical Sciences, Monash University, 381 Royal Parade, Parkville, Victoria 3052, Australia.
² School of Pharmaceutical Science, Nanjing Tech University, Nanjing, 211816, China.

PMID: 27557114
DOI: 10.4155/fmc-2016-0151

No abstract available

Keywords: histone acetyltransferase inhibitors; lysine acetyltransferase inhibitors; small-molecule epigenetic modulators.

Publication types

Editorial
Research Support, Non-U.S. Gov't

MeSH terms

Enzyme Inhibitors / chemistry
Enzyme Inhibitors / metabolism*
Epigenesis, Genetic
Histone Acetyltransferases / antagonists & inhibitors
Histone Acetyltransferases / metabolism*
Humans
Lysine Acetyltransferases / antagonists & inhibitors
Lysine Acetyltransferases / metabolism
Small Molecule Libraries / chemistry
Small Molecule Libraries / metabolism

Substances

Enzyme Inhibitors
Small Molecule Libraries
Lysine Acetyltransferases
Histone Acetyltransferases