Perspectives in Medicinal Chemistry: DNA Methylation and Demethylation Mechanisms as Therapeutic Targets?

Curr Top Med Chem. 2016;16(8):807-8. doi: 10.2174/1568026616999151013124703.
No abstract available

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Azacitidine / analogs & derivatives
  • Azacitidine / pharmacology
  • Chemistry, Pharmaceutical / methods
  • Chemistry, Pharmaceutical / trends
  • DNA Glycosylases / metabolism
  • DNA Methylation*
  • Decitabine
  • Endodeoxyribonucleases / metabolism
  • Epigenesis, Genetic
  • Humans
  • Neoplasms / drug therapy
  • Neoplasms / genetics*

Substances

  • Decitabine
  • Endodeoxyribonucleases
  • MBD4 protein, human
  • DNA Glycosylases
  • Azacitidine