Abstract
Synthetic approaches to macrosphelide derivatives, based on medicinal chemistry, are summarized. This review contains conventional medicinal chemistry approaches, combinatorial chemistry, fluorous tagging techniques and affinity chromatography preparation. In addition, advances in their apoptosis-inducing activities are also included.
Publication types
-
Research Support, Non-U.S. Gov't
-
Review
MeSH terms
-
Animals
-
Antineoplastic Agents / chemical synthesis*
-
Antineoplastic Agents / pharmacology
-
Apoptosis / drug effects*
-
Combinatorial Chemistry Techniques*
-
Drug Discovery
-
Humans
-
Macrolides / chemical synthesis*
-
Macrolides / pharmacology
Substances
-
Antineoplastic Agents
-
Macrolides