Pyrimido[4,5-d]pyrimidin-4(1H)-one derivatives as selective inhibitors of EGFR threonine790 to methionine790 (T790M) mutants

Angew Chem Int Ed Engl. 2013 Aug 5;52(32):8387-90. doi: 10.1002/anie.201302313. Epub 2013 Jun 26.
No abstract available

Keywords: T790M mutants; drug design; inhibitors; selectivity.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Cell Proliferation
  • Drug Design
  • ErbB Receptors / antagonists & inhibitors*
  • Methionine / chemistry*
  • Threonine / chemistry*

Substances

  • Threonine
  • Methionine
  • ErbB Receptors