Small molecule bromodomain inhibitors: extending the druggable genome

Prog Med Chem. 2012:51:1-55. doi: 10.1016/B978-0-12-396493-9.00001-7.
No abstract available

Publication types

  • Review

MeSH terms

  • Acetylation
  • Amino Acid Sequence
  • Animals
  • Autoimmune Diseases / drug therapy
  • Autoimmune Diseases / genetics
  • Communicable Diseases / drug therapy
  • Drug Design*
  • Epigenesis, Genetic
  • Humans
  • Metabolic Diseases / drug therapy
  • Metabolic Diseases / genetics
  • Metabolic Diseases / metabolism
  • Molecular Sequence Data
  • Neoplasms / drug therapy
  • Neoplasms / genetics
  • Protein Structure, Tertiary*
  • Proteins / antagonists & inhibitors*
  • Proteins / chemistry*
  • Proteins / genetics
  • Small Molecule Libraries

Substances

  • Proteins
  • Small Molecule Libraries