A structure-activity relationship study of the antimalarial and antileishmanial activities of nonpeptide macrocyclic histone deacetylase inhibitors

ChemMedChem. 2010 Aug 2;5(8):1232-5. doi: 10.1002/cmdc.201000087.
No abstract available

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Antimalarials / chemistry*
  • Antimalarials / pharmacology
  • Antiprotozoal Agents / chemistry*
  • Antiprotozoal Agents / pharmacology
  • Histone Deacetylase Inhibitors / chemistry*
  • Histone Deacetylase Inhibitors / pharmacology
  • Histone Deacetylases / chemistry*
  • Histone Deacetylases / metabolism
  • Leishmania / drug effects*
  • Macrocyclic Compounds / chemistry*
  • Macrocyclic Compounds / pharmacology
  • Plasmodium falciparum / drug effects
  • Structure-Activity Relationship

Substances

  • Antimalarials
  • Antiprotozoal Agents
  • Histone Deacetylase Inhibitors
  • Macrocyclic Compounds
  • Histone Deacetylases