Synthesis and insecticidal activity of N-substituted (1,3-thiazole)alkyl sulfoximine derivatives

Haibo Yu; Zhenfang Qin; Hong Dai; Xin Zhang; Xue Qin; Tingting Wang; Jianxin Fang

doi:10.1021/jf802802g

Synthesis and insecticidal activity of N-substituted (1,3-thiazole)alkyl sulfoximine derivatives

J Agric Food Chem. 2008 Dec 10;56(23):11356-60. doi: 10.1021/jf802802g.

Authors

Haibo Yu¹, Zhenfang Qin, Hong Dai, Xin Zhang, Xue Qin, Tingting Wang, Jianxin Fang

Affiliation

¹ Research Institute of Elemento-Organic Chemistry, Nankai University, Tianjin, People's Republic of China.

PMID: 19007296
DOI: 10.1021/jf802802g

Abstract

The N-substituted alkyl sulfoximine derivatives are a new chemical family of neonicotinoid insecticides. We have designed and synthesized 10 (1,3-thiazole)alkyl sulfoximine derivatives. All compounds were identified by (1)H and (13)C nuclear magnetic resonance (NMR), IR, and elemental analyses. Preliminary bioassays indicated that some title compounds exhibited good insecticidal activities at 10 mg/L against Myzus persicae . The relationship between structure and biological activity was also discussed.

Publication types

Research Support, Non-U.S. Gov't

MeSH terms

Animals
Aphids / drug effects
Insecticides / chemical synthesis
Insecticides / chemistry*
Insecticides / pharmacology*
Structure-Activity Relationship

Substances

Insecticides